Synthesis of progesterone heterocyclic derivatives of potential antimicrobial activity

F. Desarnaud, A. N. Dothi, A. M. Brown, G. Lemke, U. Suter, E. E. Baulieu and M. Schumacher, Progesterone stimulates the activity of the promoters of peripheral myelin protein-22 and protein zero genes in Schwann cells, J. Neurochem.71 (1998) 1765-1768.10.1046/j.1471-4159.1998.71041765.xSearch in Google Scholar

R. C. Melcangi, V. Magnaghi, I. Cavarretta, I. Zucchi, P. Bovolin, D. D'Urso and L. Martini, Progesterone derivatives are able to influence peripheral myelin protein-22 and P0 gene expression: possible mechanisms of action, J. Neurosci. Res.56 (1999) 349-357; DOI: 10.1002/(SICI)1097-4547(19990515).Search in Google Scholar

R. M. Mohareb, J. Z. Ho and F. E. Elfarouk, Synthesis of thiophenes, azoles and azines with potential biological activity by employing the versatile heterocyclic precursor N-benzoylcyanoacetylhydrazine, J. Chin. Chem. Soc.54 (2007) 1053-1066.10.1002/jccs.200700152Search in Google Scholar

H. Z. Shams, R. M. Mohareb, M. H. Helal and A. E. Mahmoud, Synthesis, structure elucidation, and biological evaluation of some fused and/or pendant thiophene, pyrazole, imidazole, thiazole, triazole, triazine and coumarin systems based on cyanoacetic 2-[(benzoylamino)thioxomethyl]hydrazide, Phosphorus Sulfur182 (2007) 237-263; DOI: 10.1080/1042500600892776.Search in Google Scholar

R. M. Mohareb, J. Z. Ho and A. A. Mohamed, Uses of 1-cyanoacetyl-4-phenyl-3-thiosemicarbazide in heterocyclic synthesis: Synthesis of thiazole, coumarin and pyridine derivatives with antimicrobial and antifungal activities, Phosophus Sulfur182 (2007) 1661-1681; DOI: 10.1080/10426500701289914.10.1080/10426500701289914Search in Google Scholar

IUPAC, Joint Commission on Biochemical Nomenclature (JCBN), Nomenclature of Steroids, Pure Appl. Chem.61 (1989) 1783-1822.10.1351/pac198961101783Search in Google Scholar

IUPAC, Joint Commission on Biochemical Nomenclature (JCBN), The Nomenclature of Steroids, Recommendations (1989), Eur. J. Biochem.186 (1989) 429-458.10.1111/j.1432-1033.1989.tb15228.xSearch in Google Scholar

O. Abdelhamid, M. M. Abdelhalim and G. A. Elmegeed, New routes to steroidal heterocyclic derivatives: synthesis of biologically active pyrazol- and isoxazolylpregnene derivatives, J. Heterocyclic Chem.44 (2007) 7-11.Search in Google Scholar

P. M. Hawkey and A. A. Lewis, Medical Bacteriology - A Practical Approach, Oxford University Press, Oxford 1994, pp. 181-194.Search in Google Scholar

N. Rameshkumar, M. Ashokkumar, E. H. Subramanian, E. R. Ilavarasan and S. K. Sridhar, Synthesis of 6-flouro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid derivatives as potential antimicrobial agents, Eur. J. Med. Chem.38 (2003) 1001-1004; DOI: 10.1016/S0223-5234(03)00151.Search in Google Scholar

R. M. Mohareb, R. A. Ibrahim and J. Z. Ho, The reaction of cyanoacetylhydrazine with ω-bromoacetophenone: Novel synthesis of 1,3,4-oxadiazine, pyridazine and coumarin derivatives, J. Chil. Chem. Soc.52 (2007) 1076-1081.Search in Google Scholar

Archana, V. K. Srivastava and A. Kumar, Synthesis of newer thiadiazolyl and thiazolidinonyl quinazolin-4(3H)-ones as potential anticonvulsant agents, Eur. J. Med. Chem.37 (2002) 873-882; DOI: 10.1016/S0223-5234(02)01389-2.10.1016/S0223-5234(02)01389-2Search in Google Scholar

D. I. Brahmbhatt, S. Shashibala and K. C. Patel, Characterization and biological activity of some polycoumarin ethylenes, Eur. Polymer J.35 (1999) 317-324; DOI: 101016/ Chodankar and S. Seshadri, Absorption-emission spectra studies of 3-hetarylcoumarin, Dyes S0014-3057(98)00127.Search in Google Scholar

N. K. Chodankar and S. Seshadri, Absorption-emission spectra studies of 3-hetarylcoumarin, Dyes Pigments6 (1984) 331-340.10.1016/0143-7208(85)85003-8Search in Google Scholar