Open Access

Some variables affecting the characteristics of Eudragit E-sodium alginate polyelectrolyte complex as a tablet matrix for diltiazem hydrochloride

1. V. A. Kemenova, R. I. Moustafine, K. V. Alekseyev, A. M. Scorodinskaya, A. B. Zezin, A. I. Tencova and V. A. Kabanov, Applying interpolymer complexes in pharmacy, Pharmacia 60 (1991) 67-72.Search in Google Scholar

2. E. Tsuchida and K. Abe, Interactions between macromolecules in solution and intermacromolecular complexes, Adv. Polym. Sci. 45 (1982) 1-147; DOI: 10.1007/BFb0017548.10.1007/BFb0017548Search in Google Scholar

3. B. Philipp, H. Dautzenberg, K. J. Linow, J. Koetz and W. Dawydoff, Polyelectrolyte complexes- -recent developments and open problems, Progr. Polym. Sci. 14 (1989) 91-172; DOI: 10.1016/ 0079-6700(89)90018-X.10.1016/0079-6700(89)90018-XSearch in Google Scholar

4. J. Koetz, H. Koepke, G. Schmidt-Naake and O. Vogl, Polyanion-polycation complex formation as a function of the position of the functional groups, Polymer 37 (1996) 2775-2781; DOI: 10.1016/ 0032-3861(96)87641-5.10.1016/0032-3861(96)87641-5Search in Google Scholar

5. S. Dumitriu and E. Chornet, Inclusion and release of proteins from polysaccharide-based polyion complexes, Adv. Drug Deliv. Rev. 31 (1998) 223-246; DOI: 10.1016/S0169-409X(97)00120-8.10.1016/S0169-409X(97)00120-8Search in Google Scholar

6. G. Dhanuja, B. Smitha and S. Sridhar, Pervaporation of isopropanol-water mixtures through polyion complex membranes, Sep. Purif. Technol. 44 (2005) 130-138; DOI: 10.1016/j.seppur.2005. 01.001.Search in Google Scholar

7. C. Tapia, E. Costa, M. Moris, J. Sapag-Hagar, F. Valenzuela and C. Basualto, Study of the influence of the pH media dissolution, degree of polymerization and degree of swelling of the polymers on the mechanism of release of diltiazem from matrices based on mixtures of chitosan/ alginate, Drug Dev. Ind. Pharm. 28 (2002) 217-224; DOI: 10.1081/DDC-120002455.10.1081/DDC-120002455Search in Google Scholar

8. R. K. Chang, Y. Peng, N. Trivedi and A. J. Shukla, Polymethacrylate, in Handbook of Pharmaceutical Excipients (Ed. R. C. Rowe, P. J. Sheskey and M. E Quinn), Pharmaceutical Press and American Pharmacists Association, USA 2009, pp. 525-533.Search in Google Scholar

9. S. K. Bajpai and S. Shubhra, Investigation of swelling/degradation behaviour of alginate beads crosslinked with Ca2+ and Ba2+ ions, Reac. Func. Poly. 59 (2004) 129-140; DOI: 10.1016/ j.reactfunctpolym.2004.01.002.10.1016/j.reactfunctpolym.2004.01.002Search in Google Scholar

10. S. Takka and F. Acartürk, Calcium alginate microparticles for oral administration: I-Effect of sodium alginate type on drug release and drug entrapment efficiency, J. Microencapsul. 16 (1999) 275-290; DOI: 10.1080/026520499289013.10.1080/02652049928901310340214Search in Google Scholar

11. C. V. Liew, L. W. Chan, A. L. Ching and P. W. Heng, Evaluation of sodium alginate as drug release modifier in matrix tablets, Int. J. Pharm. 309 (2006) 25-37; DOI: 0.1016/j.ijpharm.2005. 10.040.10.1016/j.ijpharm.2005.10.04016364576Search in Google Scholar

12. Martindale: The Complete Drug Reference (Ed. P. Kathleen), 35th ed., The Pharmaceutical Press, London 2007, pp. 1136-1138.Search in Google Scholar

13. R. I. Moustafine, I. M. Zaharov and V. A. Kemenova, Physicochemical and drug release properties of Eudragit®E PO/Eudragit®L 100-55 interpolyelectrolyte complexes, Eur. J. Pharmac. Biopharmac. 63 (2006) 26-36; DOI: 10.1016/j.ejpb.2005.10.005.10.1016/j.ejpb.2005.10.00516380241Search in Google Scholar

14. H. J. Prado, M. C. Matulewicz, P. Bonelli and A. L. Cukierman, Basic butylated methacrylate copolymer/ kappa-carrageenan interpolyelectrolyte complex: Preparation, characterization and drug release behaviour, Eur. J. Pharmac. Biopharmac. 70 (2008) 171-178; DOI: 10.1016/j.ejpb.2008.04.017.10.1016/j.ejpb.2008.04.01718583115Search in Google Scholar

15. A. Bani-Jaber, L. Al-Aani, H. Alkhatib and B. Al-Khalidi, Prolonged intragastric drug delivery mediated by Eudragit® E-carrageenan, polyelectrolyte matrix tablets, AAPS Pharm. Sci. Tech. 12 (2011) 354-361; DOI: 10.1208/s12249-011-9595-0.10.1208/s12249-011-9595-0Search in Google Scholar

16. A. H. Abd El-Gawad, E. M. Ramadan, O. A. Soliman and R. M. Yusif, Formulation and in-vivo study of diltiazem hydrochloride tablets prepared using interpolymer complexes, BJPR 2 (2012) 17-40.10.9734/BJPR/2014/1049Search in Google Scholar

17. R. W. Korsmeyer, R. Gurny, E. M. Doelker, P. Buri and N. A. Peppas, Mechanism of solute release from porous hydrophilic polymers, Int. J. Pharm. 15 (1983) 25-35; DOI: 10.1016/0378-5173 (83)90064-9.Search in Google Scholar

18. R. I. Moustafine, V. A. Kemenova, and G. Van den Mooter, Characteristics of interpolyelectrolyte complexes of Eudragit E100 with sodium alginate, Int. J. Pharm. 294 (2005) 113-120; DOI: 10.1016/j.ijpharm.2005.01.029.10.1016/j.ijpharm.2005.01.029Search in Google Scholar

19. J. P. Soares, J. E. Santos, G. O. Chierice and ETG Cavalheiro, Thermal behavior of alginic acid and its sodium salt, Eclet Quim. 29 (2004) 57-64; DOI: 10.1590/S0100-46702004000200009.10.1590/S0100-46702004000200009Search in Google Scholar

20. S. Y. Lin, H. L. Yu and M. J. Li, Formation of six-membered cyclic anhydrides by thermally induced intramolecular ester condensation in Eudragit E film, Polymer 40 (1999) 3589-3593; DOI: 10.1016/S0032-3861(98)00488-1.10.1016/S0032-3861(98)00488-1Search in Google Scholar

21. K. Saeio, Y. Pongpaibul, H. Vierstein and S. Okonogi, Factors influencing drug dissolution characteristic from hydrophilic polymer matrix tablet, Sci. Pharm. 75 (2007) 147-163; DOI: 10.3797/ scipharm.2007.75.147.10.3797/scipharm.2007.75.147Search in Google Scholar

22. V. M. Rao, K. Engh and Y. Qiu, Design of pH-independent controlled release matrix tablets for acidic drugs, Int. J. Pharm. 252 (2003) 81-86; DOI: 10.1016/S0378-5173(02)00622-1.10.1016/S0378-5173(02)00622-1Search in Google Scholar

23. W. M. Obeidat, A. H. Abuznait and A. S. Sallam, Sustained release tablets containing soluble polymethacrylates: Comparison with tableted polymethacrylate IPEC polymers, AAPS Pharm. Sci. Tech. 11 (2010) 54-63; DOI: 10.1208/s12249-009-9348-5.10.1208/s12249-009-9348-5Search in Google Scholar

24. M. E. C. Aldrete and L. V. Robles, Influence of the viscosity grade and particle size of HPMC on metronidazole release from matrix tablets, Eur. J. Pharmac. Biopharmac. 43 (1997) 173-178; DOI: 10.1016/S0939-6411(96)00004-5.10.1016/S0939-6411(96)00004-5Search in Google Scholar

25. J. Siepmann, H. Kranz, R. Bodmeier and N. A. Peppas, HPMC-matrices for controlled drug delivery: a new model combining diffusion, swelling and dissolution mechanisms and predicting the release kinetics, Pharm. Res. 16 (1999) 1748-1756; DOI: 10.1023/A:1018914301328.10.1023/A:1018914301328Search in Google Scholar

26. C. Tapia, Z. Escobar, E. Costa, J. S. Hagar, F. Valenzuela, C. Basualto, M. N. Gai and M. Y. Pedram, Comparative studies on polyelectrolyte complexes and mixtures of chitosan-alginate and chitosan-carrageenan as prolonged diltiazem chlorhydrate release systems, Eur. J. Pharmac. Biopharmac. 57 (2004) 65-75; DOI: 10.1016/S0939-6411(03)00153-X.10.1016/S0939-6411(03)00153-XSearch in Google Scholar

27. H. M. Fahmy and M. M. G. Fouda, Crosslinking of alginic acid/chitosan matrices using polycarboxylic acids and their utilization for sodium diclofenac release, Carbohyd. Polym. 73 (2008) 606-611; DOI: 10.1016/j.carbpol.2007.12.024.10.1016/j.carbpol.2007.12.02426048227Search in Google Scholar

28. K. Satoh, K. Takayama, Y. Machida, Y. Suzuki and T. Nagai, Disintegration and dissolution characteristics of compressed tablets consisting of hydroxypropyl cellulose and carboxyvinyl polymer, Chem. Pharm. Bull. 37 (1989) 1642-1644.10.1248/cpb.37.1642Search in Google Scholar

29. M. M. Talukdar, I. Vinckier, P. Moldenaers and R. Kinget, Rheological characterization of xanthan gum and hydroxypropylmethyl cellulose with respect to controlled-release drug delivery, J. Pharm. Sci. 85 (1996) 537-540; DOI: 10.1021/js950476u.10.1021/js950476u8742947Search in Google Scholar

30. D. Ray, P. S. Gils, G. P. Mohanta, R. Manavalan and P. K. Sahoo, Comparative delivery of diltiazem hydrochloride through synthesized polymer. Hydrogel and hydrogel microspheres, J. Appl. Polym. Sci. 116 (2010) 959-968; DOI: 10.1002/app.31661. 10.1002/app.31661Search in Google Scholar

eISSN:
1846-9558
ISSN:
1330-0075
Language:
English
Publication timeframe:
4 times per year
Journal Subjects:
Pharmacy, other