Search Results

You are looking at 1 - 10 of 34 items for :

Clear All
Open access

Rafat M. Mohareb, Amira E. M. Abdallah and Ebtsam A. Ahmed

References 1. I. Lagoja, C. Pannecouque, G. Griffioen, S. Wera, V. M. Rojasdelaparra and A. V. Aerschot, Substituted 2-aminothiazoles are exceptional inhibitors of neuronal degeneration in tau-driven models of Alzheimer’s disease, Eur. J. Med. Chem. 43 (2011) 386-392; https://doi.org/org/10.1016/j.ejps.2011.05.014 2. S. Kamila, K. Mendoza and E. R. Biehl, Microwave-assisted Hantzsch thiazole synthesis of Nphenyl- 4-(6-phenylimidazo[2,1-b]thiazol-5-yl)thiazol-2-amines from the reaction of 2-chloro-1-(6- phenylimidazo[2,1-b

Open access

Zita Tokárová and Anna Biathová

, Hosseinzadeh-Khanmiri R, Ghorbani-Kalhor E (2017) N-Propargylamines: versatile building blocks in the construction of thiazole cores. Belst. J. Org. Chem. 13: 625-638. Beno BR, Yeung K-S, Bartberger MD, Pennington LD, Meanwell NA, (2015) A survey of the role of noncovalent sulfur interactions in drug design. J. Med. Chem. 58: 4383-4438. Bevk D, Marin L, Lutsen L, Vanderzande D, Maes W (2013) Thiazolo[5,4-d]thiazoles - promising building blocks in the synthesis of semiconductors for plastic electronics (Review). RSC Adv. 3: 11418

Open access

Mostafa M. Ghorab, Mansour S. Alsaid, Mohammed S. Al-Dosari, Fatma A. Ragab, Abdullah A. Al-Mishari and Abdulaziz N. Almoqbil

of new drug molecules to be used in reversing multidrug resistance in cancer, Curr. Cancer Drug Targets 9 (2009) 298–306; DOI: 10.2174/156800909788166619. 6. M. G. Ferlin, B. Gatto, G. Chiarelotto and M. Palumbo, Pyrroloquinoline derivatives as potential antineoplastic drugs, Bioorg. Med. Chem. 8 (2000) 1415–1422; DOI: 10.1016/S0968-0896(00)00060-2. 7. M. S. Alsaid, M. S. Bashandy, S. I. Al-Qasoumi and M. M. Ghorab, Anti-breast cancer activity of some novel 1,2-dihydropyridine, thiophene and thiazole derivatives, Eur. J. Med. Chem. 46 (2011

Open access

Mohammed Albratty, Karam Ahmed El-Sharkawy and Hassan Ahmed Alhazmi

antioxidant activity of 1,3,4-oxadiazole tagged thieno[2,3- d ]pyrimidine derivatives, Eur. J. Med. Chem . 58 (2012) 340–345; https://doi.org/10.1016/j.ejmech.2012.10.007 7. N. C. Desai, N. Bhatt, H. Somani and A. Trivedi, Synthesis, antimicrobial and cytotoxic activities of some novel thiazole clubbed 1,3,4-oxadiazoles, Eur. J. Med. Chem . 67 (2013) 54–59; https://doi.org/10.1016/j.ejmech.2013.06.029 8. M. Mahesh, G. Bheemaraju, G. Manjunath and P. V. Ramana, Synthesis of new oxadiazole, pyrazole and pyrazolin-5-one bearing 2-((4-methyl-2-oxo-2 H -chromen-7-yl

Open access

Lulzime Ballazhi, Emil Popovski, Ahmed Jashari, Faik Imeri, Ibrahim Ibrahimi, Bozhana Mikhova and Kristina Mladenovska

, Synthesis and primary cytotoxicity evaluation of new imidazo[ 2,1-b]thiazole derivatives, Eur. J. Med. Chem. 42 (2007) 320-326; DOI: 10.1016/j.ejmech. 2006.10.012. 22. M. J. Choi, E. S. No, D. A. Thorat, J. W. Jang, H. Yang, J. Lee, H. Choo, S. J. Kim, C. S. Lee, S. Y. Ko, J. Lee, G. Nam and A. N. Pae, Synthesis and biological evaluation of aryloxazole derivatives as antimitotic and vascular-disrupting agents for cancer therapy, J. Med. Chem. 56 (2013) 9008-9018; DOI: 10.1021/jm400840p. 23. P. Poma, M. Notarbartolo, M. Labbozze_ a, A

Open access

M. Żmigrodzka, M. Guzera and A. Winnicka

) Demonstration that thiazole-orange-positive platelets in the dog are less than 24 hours old. Blood 85: 1822-1825. Davis B, Toivio-Kinnucan M, Schuller S, Boudreaux MK (2008) Mutation in beta-tubulin correlates with macrothrombocytopenia in Cavalier King Charles Spaniels. J Vet Intern Med 22: 540-545. Harrison P (1998) Reticulated platelets. CME Bull Haematol 2: 43-45. Ingram M, Coopersmith A (1969) Reticulated platelets following acute blood loss. Br J Haematol 17: 225-229. Kienast J, Schmitz G (1990) Flow

Open access

Mostafa M. Ghorab, Mahmoud S. Bashandy and Mansour S. Alsaid

. Khalil, M. A. Berghot and M. A. Gouda, Synthesis and antibacterial activity of some new thiazole and thiophene derivatives, Eur. J. Med. Chem. 44 (2009) 4434-4440; DOI: 10.1016/j.ejmech. 2009.06.002. 4. S. Deka, S. Mohan, J. Saravanan, M. Kakati, A. Talukdar, B. J. Sahariah, B. K. Dey and R. K. Sarma, Syntheses, characterization and in-vitro anti-Inflammatory activity of some novel thiophenes, Maced. J. Med. Sci. 5 (2012) 159-163; DOI: org/10.3889/MJMS.1957-5773.2012.0225. 5. R. A. Forsch, J. E. Wright and A. Rosowsky, Synthesis and in

Open access

Rafat Mohareb and Hanaa Hana

(1999) 349-357; DOI: 10.1002/(SICI)1097-4547(19990515). R. M. Mohareb, J. Z. Ho and F. E. Elfarouk, Synthesis of thiophenes, azoles and azines with potential biological activity by employing the versatile heterocyclic precursor N -benzoylcyanoacetylhydrazine, J. Chin. Chem. Soc. 54 (2007) 1053-1066. H. Z. Shams, R. M. Mohareb, M. H. Helal and A. E. Mahmoud, Synthesis, structure elucidation, and biological evaluation of some fused and/or pendant thiophene, pyrazole, imidazole, thiazole, triazole, triazine and

Open access

J. Višņevska, E. Jaščenko, I. Šestakova, A. Gulbe and E. Ābele

References Moody, C. J., Roffey, J. R., Stephens, M. A., Stratford, I. J. (1997). Synthesis and cytotoxic activity of indolyl thiazoles. Antitumor Drugs, 8 (5), 489-499. Kumar, R., Lown, J. W. (2003). Synthesis and antitumor cytotoxicity evaluation of novel thiazole-containing glycosylated polyamides. Eur J. Org. Chem. , (24), 4842-4851. Lu, Y., Li, C.-M., Wang, Z., Ross, C. R., Chen, J., Dalton, J., Li, W., Miller, D. D. (2009). Discovery of 4-substituted methoxybenzoyl

Open access

Rafat M. Mohareb, Amira E. M. Abdallah, Maher H. E. Helal and Somiya M. H. Shaloof

benzothiophene cell activation inhibitor, Toxicology 98 (1995) 111–123; DOI: 10.1016/0300-483X(94)02985-4. 15. H. Z. Shams, R. M. Mohareb, M. H. Helal and A. E. Mahmoud, Synthesis, structure elucidation, and biological evaluation of some fused and/or pendant thiophene, pyrazole, imidazole, thiazole, triazole, triazine, and coumarin systems based on cyanoacetic 2-[(benzoylamino)thioxomethyl] hydrazide, Phosphorus Sulfur Silicon 182 (2007) 237–263; DOI: 10.1080/10426500600892776. 16. L. Berrade, B. Aisa, M. J. Ramirez, S. Galiano, S. Guccione, L. R. Moltzau