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Khushal M. Kapadiya, Yashwantsinh S. Jadeja, Avishek Banik and Ranjan C. Khunt

, Thakrar S, et al. Synthesis and biological evaluation of 4-styrylcoumarin derivatives as inhibitors of TNF-a and IL-6 with anti-tubercular activity. Bioorg Med Chem Lett 2011;21(8):2547-9. 13. Khunt R, Khedkar V, Coutinho E. Synthesis and 3D-QSAR analysis of 2-chloroquinoline derivatives as H37RV MTB inhibitors. Chem Biol Drug Des 2013;82:669. 14. De Boer RA, Voors AA, Van Veldhuisen DJ. Nebivolol: third-generation beta-blockade. Expert Opin Pharmacother 2007;8(10):1539-50. 15. Grundner C, Ng Hl, Alber T. Mycobacterium tuberculosis protein tyrosine

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Dan-Dan Zhang, Pi Luo, Ying Chen, Zheng-Feng Wang, Wan-Hui Ye and Hong-Lin Cao

. SKALETSKY (2000): Primer3 on the WWW for general users and for biologist programmers, pp. 365-386. In: Methods in molecular biology, vol. 132: Bioinformatics methods and protocols, edited by S. MISENER and S. A. KRAWETZ, Humana Press, Totowa, New Jersey, USA. WU, C. C., C. F. PENG, I. L. TSAI, M. H. ABD EL-RAZEK, H. S. HUANG and I. S. CHEN (2007): Secondary metabolites from the roots of Engelhardia roxburghiana and their antitubercular activities. Phytochemistry 68: 1338-1343. WU, H. C., M. J. CHENG, C. F. PENG, S. C. YANG, H. S. CHANG, C

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Ivana Zemanová and Renata Gašparová

., LOURENCO, C.S.M., CALVALHO, S.L.G., ALMEIDA, C.B.M, CUNHA, C.A.: Synthesis, antitubercular activity, and SAR study of N-substitutedphenylamino-5-methyl-1H-1,2,3-triazole-4-carbohydrazides. Bioorg. Med. Chem., 19, 2011, 5605-5611. KRUTOŠÍKOVÁ, A., DANDÁROVÁ, M., ALFÖLDI, J.: Synthesis and reactions of furo[3,2- b ]pyrrole type aldehydes. Coll. Czech. Chem. Commun., 58, 1993, 2139-2149. KRUTOŠÍKOVÁ, A., DANDÁROVÁ, M., ALFÖLDI, J.: Substituted vinyl azides in the synthesis of condensed nitrogen heterocycles. Chem. Papers, 48, 1994, 268

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Satyajit Dutta

)methyl)-quinazoline-4(3 H )-one and their derivatives for anti-tubercular activity, Indian J. Chem.   45B (2006) 1778-1781. P. Gupta, S. Hameed and R. Jain, Ring-substituted imidazoles as a new class of anti-tuberculosis agents, Eur. J. Med. Chem.   39 (2004) 805-814; DOI: 10.1016/j.cjmech.2004.05.005. V. Alagarsamy, R. Giridhar, M. R. Yadav, R. Revathi, K. Ruckmani and E. De Clercq, Anti HIV, antibacterial, and antifungal activities of some novel 1,4-disubstituted-1,2,4-triazolo [4,3- a ]quinazolin-5(4 H )-ones, Indian J

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Priya V. Frank, Mahesha Manjunatha Poojary, Naral Damodara and Chandrashekhar Chikkanna

-thione derivatives: Promising anticancer agents, Bioorg. Med. Chem . 14 (2006) 1236-1246; DOI: 10.1016/j.bmc.2005.09.053. 4. M. A. Ali and M. Shaharyar, Oxadiazole Mannich bases: Synthesis and antimycobacterial activity, Bioorg. Med. Chem . Lett. 17 (2007) 3314-3316; DOI: 10.1016/j.bmcl.2007.04.004. 5. D. Sriram, D. Banerjee and P. Yogeeshwari, Efavirenz Mannich bases: Synthesis, anti-HIV and antitubercular activities, J. Enzyme Inhib. Med. Chem. 24 (2009) 1-5; DOI: 10.1080/14756360701404159. 6. B. M. Kotecka, G

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Saleh A. Bahashwan

REFERENCES 1. A. B. Siddiqui, A. R. Trivedi, V. B. Kataria and V. H. Shah, 4,5-Dihydro-1 H -pyrazolo[3,4- d ]pyrimidine containing phenothiazines as antitubercular agents, Bioorg. Med. Chem. Lett. 51 (2014) 1493–1495; DOI: 10.1016/j.bmcl.2014.02.012. 2. N. M. Y. Elsayed, D. A. Abou El Ella, R. A. T. Serya, M. F. Tolba, R. Shalaby and K. A. M. Abouzid, Design, synthesis and biological evaluation of indazole-pyrimidine based derivatives as anticancer agents with anti-angiogenic and antiproliferative activities, Med. Chem. Commun. 7 (2016) 881

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Mohammed Albratty, Karam Ahmed El-Sharkawy and Shamsher Alam

- sulfonylthiophenes and related compounds as a new class of diarylsulfones, Bioorg. Med. Chem. 9 (2001) 1123-1132; DOI: 10.1016/S0968-0896(00)00333-3. 4. S. Sulzer-Mosse, F. Cederbaum, C. Lamberth, G. Berthon, J. Umarye, V. Grasso, A. Schlereth, M. Blum and R. Waldmeier, Synthesis and fungicidal activity of N-thiazol-4-yl-salicylamides, a new family of anti-oomycete compounds, Bioorg. Med. Chem. 23 (2015) 2129-2138; DOI: 10.1016/j. bmc.2015.03.007. 5. V. Padmavathi, C. Prema Kumari, B. C. Venkatesh and A. Padmaja, Synthesis and

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Mohammed Albratty, Karam Ahmed El-Sharkawy and Hassan Ahmed Alhazmi

REFERENCES 1. N. C. Desai, H. Somani, A. Trivedi, K. Bhatt, L. Nawale, V. M. Khedkar, P. C. Jha and D. Sarkar, Synthesis, biological evaluation and molecular docking study of some novel indole and pyridine based 1,3,4-oxadiazole derivatives as potential antitubercular agents, Bioorg. Med. Chem. Lett . 26 (2016) 1776–1783; https://doi.org/10.1016/j.bmcl.2016.02.043 2. A. G. Banerjee, N. Das, S. A. Shengule, R. S. Srivastava and S. K. Shrivastava, Synthesis, characterization, evaluation and molecular dynamics studies of 5,6-diphenyl-1,2,4-triazin-3(2 H

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Peter O. Osarumwense

, Indian Journal of Chemistry 48B (2009) 840- 47. [10]. P. Paneersalvam, T. Raj, M.P.S. Ishar, B. Singh, V. Sharma, B.A. Rather, Anticonvulsant activity of Schiff bases of 3-amino - 6, 8 -dibromo - 2 - phenyl - quinazolin - 4(3H) - ones, Indian Journal of Pharmaceutical Sciences 72 (2010) 375 - 378. Doi: 10.4103/0250-474X.70488 70488 [11]. P. Nandy, M.T. Vishalakshi, A.R. Bhat, Synthesis and antitubercular activity of Mannich bases of 2-methyl-3H-quinazolin-4-ones, Indian Journal of Heterocyclic Chemistry 15 (2006) 293 - 294

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Eman M. Flefel, Randa E. Abdel-Mageid, Waled A. Tantawy, Mohamed A. Ali and Abd El-Galil E. Amr

0201677. 12. G. V. S. Kumar, Y. Rajendraprasad, B. P. Mallikarjuna, S. M. Chandrashekar and C. Kistayya, Synthesis of some novel 2-substituted-5-[isopropylthiazole clubbed] 1,2,4-triazole and 1,3,4-oxadiazoles as potential antimicrobial and antitubercular agents , Eur. J. Med. Chem. 45 (2010) 2063-2074; DOI: 10.1016/j.ejmech.2010.01.045. 13. K. Imtiaz, A. Sajid, H. Shahid, H. R. Nasim, T. H. Muhammad, W. Abdul, U. Reaz, U. Zaheer, K. Ajmal, A. M. Sajjad and C. Iqbal, Synthesis, antioxidant activities and urease inhibition of some new 1