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Pharmacokinetics of cytisine after single intravenous and oral administration in rabbits

derivatives and of bioisosteric thiocytisine as potent and selective nAChR ligands. Eur J Med Chem   36 : 375-388. Jorenby D, Hays J, Rigotti N, Azoulay S, Watsky E, Williams K, Billing C, Gong J and Reeves K. (2006). Efficacy of varenicline, an α 4 β 2 -nicotinic acetylcholine receptor partial agonist, vs. placebo or sustained-release bupropion for smoking cessation. A randomized controlled trial. JAMA   296 : 56-63. Klocking H, Richter M, and Damm G. (1980). Pharmacokinetic studies with 3 Hcytisine. Arch Toxicol

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Interdisciplinary Toxicology
The Journal of Institute of Experimental Pharmacology of Slovak Academy of Sciences
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Comparison of oral bioavailability of acetaminophen tablets, capsules and effervescent dosage forms in healthy volunteers

.: Pharmacokinetics of paracetamol (acetaminophen) after intravenous and oral administration. Eur J Clin Pharm. 1977;11:283. 9. Srinath K, et al.: Formulation and evaluation of effervescent tablets of paracetamol. INT J Pharm Res Dev. 2011;3:76. 10. Blagden N, et al.: Crystal engineering of active pharmaceutical ingredients to improve solubility and dissolution rates. Adv Drug Deliv Rev 2007 Jul 30;59(7):617-30 Epub 2007 May 29. 11. De Silva L, et al.: Usability of mobile technology to screen for drugdrug interactions in kidney transplant patients. Am J Nephrol

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Effects of teicoplanin on cell number of cultured cell lines

REFERENCES Bibler MR, Peter TF, Hagler DN, Bode RB, Staneck JL, Thamlikitkul V. (1987). Clinical evaluation of efficacy, pharmacokinetics, and safety of teicoplanin for serious Gram-positive infections. Antimicrob Agents Chemother 31 : 207–212. Eggleston M, Ofosu J. (1988). Teicoplanin, a new agent for gram positive bacterial infection. Infect Control Hosp Epidemiol 9 : 209–211. Glupezynski Y, Lagast H, Auwera PV, Thys JP, Crokaert F, Yourassowsky E, Meunier-Carpentier F, Klastersky J, Kains JP, Serruys-Schoutens E. (1986). Clinical

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Investigation of in vitro effects of ethephon and chlorpyrifos, either alone or in combination, on rat intestinal muscle contraction

Activity in Adult Rats: An in Vitro and in Vivo Comparison. Fundam App Toxicol   38 : 148-157. Cochran RC. (2002). Appraisal of Risks from Nonoccupational Exposure to Chlorpyrifos. Reg Toxicol Pharmacol   35 : 105-121. Cook TJ and Shenoy SS. (2003). Intestinal permeability of chlorpyrifos using the single-pass intestinal perfusion method in the rat. Toxicology   184 : 125-133. El-Masri HA, Mumtaz MM and Yushak ML. (2004). Application of physiologically-based pharmacokinetic modeling to

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Synthesis and biological evaluation of some novel 1-substituted fentanyl analogs in Swiss albino mice

SW, Lai J, Porreca F, Vardanyan R, Hruby VJ. (2007). Understanding the structural requirements of 4-anilidopiperidine analogues for biological activities at mu and delta opioid receptors. Bioorg Med Chem Lett 17: 2161-2165. Lemmens H. (1995). Pharmacokinetic-pharmacodynamic relationships for opioids in balanced anaesthesia. Clin Pharmacokinet 29: 231-242. Litchfi eld JTJr, Wilcoxon F. (1949). A simplifi ed method of evaluating dose-effect experiments. J Pharm Exp Ther 96: 99-113. Mather LE. (1983). Clinical

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Distribution of opiate alkaloids in brain tissue of experimental animals

-induced analgesia: activational and organizational effects. Pharmacol Exp Ther 300: 695-701. Craft R, Heideman L, Bartok R. (1998). effect of gonadectomy on discriminative stimulus effects of morphine in female versus male rats. Drug Alcohol Depend 53: 95-109. Djurendic-Brenesel M, Mimica-Dukic N, Pilija V, Tasic M. (2010). Gender-related differences in the pharmacokinetics of opiates. Forensic Sci Int 194(1-3): 28-33. Erdtmann-Vourliotis M, Mayer P, Riechert U, Grecksch G, Höllt V. (1998). Identification of brain regions

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Effect of cytisine on some brain and hepatic biochemical parameters in spontaneously hypertensive rats

pharmacokinetic studies on nicotine, cytisine and lobeline. Neuropharmacology   29 : 619-624. Tabex. Product monograph, Sopharma, 2006. Tzankova V and Danchev N. (2007) Cytisine - from ethomedical use to the development as a natural alternative for smoking cessation. Biotechnol & Biotechnol EQ   21 : 151-160. Yoshimoto K, Komura S, Hattori H, Yamori Y, Miura A, Yoshida T, Hioki C, Kato B, Fukuda F, Tanaka S, Hirai A, Nishimura A, Sawai Y and Yashuhara M. (2003) Pharmacological studies of alcohol

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Pixantrone, a new anticancer drug with the same old cardiac problems? An in vitro study with differentiated and non-differentiated H9c2 cells

toxicity: the cardiac susceptibility to oxidative stress. Chem Res Toxicol 26 : 1285–1311. Costa VM, Silva R, Tavares LC, Vitorino R, Amado F, Carvalho F, Bastos ML, Carvalho M, Carvalho RA, Remiao F. (2009). Adrenaline and reactive oxygen species elicit proteome and energetic metabolism modifications in freshly isolated rat cardiomyocytes. Toxicology 260 : 84–96. Dawson LK, Jodrell DI, Bowman A, Rye R, Byrne B, Bernareggi A, Camboni G, Smyth JF. (2000). A clinical phase I and pharmacokinetic study of BBR 2778, a novel anthracenedione analogue

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Trends in vascular pharmacology research in the Department of Pharmacology and Clinical Pharmacology, Faculty of Medicine, Comenius University, Bratislava

, Kriška M, Kovalčík V. (1978). Bayliss myogenic response in the isolated ductus arteriosus of guinea-pig and rabbit fetuses. Experientia   34 : 745-746. Turnheim K. (2003). When drug therapy gets old: pharmacokinetics and pharmacodynamics in the elderly. Exp Gerontol   38 : 843-853. Varga Z, Kriška M, Kristová V, Hudec. (2010). Prescription of NSAIDs and risk of cardiovascular adverse effects in hospitalized patients. Rheumatologia 24 : 87-90. Vojtko R., Villaris R., Petrová M., Líšková S

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